Parameter | Unit | IV | PO |
---|---|---|---|
T1/2β | h | 6.11 ± 1.97 | 8.21 ± 2.31 |
Tmax | h | — | 0.44 ± 0.16 |
Cmax | μg/mL | — | 2.03 ± 0.73 |
AUC0-24 h | μg/mL · h | 8.43 ± 1.06 | 8.26 ± 1.08 |
VZ | L/kg | 10.4 ± 3.32 | — |
Cl | L/kg · h | 1.18 ± 0.16 | — |
VZ/F | L/kg | — | 14.1 ± 3.55 |
Cl/F | L/kg · h | — | 1.21 ± 0.17 |
MRT0-24 h | h | 4.17 ± 1.04 | 7.75 ± 1.86 |
F | % | — | 97.6 ± 5.32 |