PK parameter | SC 0.05 mg/kg [mean (SD) range] | IM 0.05 mg/kg [mean (SD) range] | IV 0.05 mg/kg [mean (SD) range] |
---|---|---|---|
Cmax/C0 (ng/mL) | 2.2 (1.4) 0.78–5.15 | 11 (3.2) 6.49–15.4*** | 71 (44) 18–169 |
F (%) | 50 (19) 26–82 | 95 (21) 53–113** | – |
t½ (min) | 260 (120) 138–495 | 148 (26) 113–191** | 139 (33) 103–197** |
tmax (min) | 39 (60) 5–180 | 11 (5) 5–15 | – |