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Table 5 Carprofen concentration measurements of plasma samples Group 6 (CA)

From: Preliminary study on carprofen concentration measurements after transcutaneous treatment with Vetdrop® in a microfracture joint defect model in sheep

Timepoint

5202 (CA) c(ng/ml)

5217 (CA) c(ng/ml)

Day 1 (day of surgery)

0.0

0.0

10 min. after 1st injection (day 1)

37500

39950

1 h after 1st injection (day 1)

29400

34217

2 h after 1st injection (day 1)

24400

27300

3 h after 1st injection (day 1)

23000

25917

12 h after 1st injection (day 1)

18200

23317

5 min prior to 2nd injection (day 2)

14100

21965

10 min after 2nd injection (day 2)

39100

43583

1 h after 2nd injection (day 2)

16000

38217

2 h after 2nd injection (day 2)

31400

37068

3 h after 2nd injection (day 2)

29200

35967

12 h after 2nd injection (day 2)

25900

31900

5 min prior to 3rd injection (day 3)

20000

25550

10 min after 3rd injection (day 3)

39700

42083

1 h after 3rd injection (day 3)

36100

40150

2 h after 3rd injection (day 3)

31900

36400

3 h after 3rd injection (day 3)

30100

34317

12 h after 3rd injection (day 3)

26200

31650

5 min prior to 4th injection (day 4)

 

27417

10 min after 4th injection (day 4)

 

41300

1 h after 4th injection (day 4)

 

39267

2 h after 4th injection (day 4)

 

37433

3 h after 4th injection (day 4)

 

36917

12 h after 4th injection (day 4)

 

32950

1 day after the last injection (day 5)

16200

23150

3 days after the last injection (day 8)

5200

6917

1 week after the last injection (day 12)

500

2115